and KCNQ1) as well as no activity on GABA(A) gated channels at 10 μM
The 30 mg/kg Amitifadine dose significantly reduces nicotine self-administration
TAME at concentration of 1-200 μM arrests interphase extract treated with recombinant cyclin B1/Cdc2 complex in mitosis
a potent muscarinic receptor agonist
GLP-1R Antagonist 1 oxy-PEG2-alcohol and KCNQ1) as well asGLP 1R Antagonist 1 (compound 5d) is an orally active, CNS penetrant and non competitive antagonist of glucagon like peptide 1 receptor (GLP 1R), with an IC50 of 650 nM. Product information CAS Number: 488097 06 9 Molecular Weight: 440. 73 Formula: C16H11ClF6N4O2 Chemical Name: 7 (4 chlorophenyl) 1,3 dimethyl 5,5 bis(trifluoromethyl) 1H,2H,3H,4H,5H,8H [1,3]diazino[4,5 d]pyrimidine 2,4 dione Smiles: